SCHEMBL8333199

SCHEMBL8333199

CCOC(=O)c1ccc(C#Cc2cc3c(cc2OC)SC(C)(C)CC3OS(=O)(=O)C(F)(F)F)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.35
CYP3A4 P08684 1/20 0.35
RARA P10276 1/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
MMP13 P45452 1/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 1/20 0.33
HSD17B2 P37059 1/20 0.33
MAPT P10636 5/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
ALDH1A1 P00352 2/20 0.31
PRKCA P17252 1/20 0.31
HTT P42858 1/20 0.31
MAPK1 P28482 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329437 0.91 MAPT (0.34) KMT2ACYP3A4RARARARBRARG
SCHEMBL6592969 0.77 NPC1 (0.36) KMT2ACYP3A4RARARARBRARG
SCHEMBL6591370 0.73 KMT2A (0.41) KMT2ACYP3A4RARARARBRARG
SCHEMBL7131831 0.70 RARA (0.36) KMT2ACYP3A4RARARARBRARG
SCHEMBL1140980 0.70 RARA (0.39) KMT2ACYP3A4RARARARBRARG
SCHEMBL727818 0.67 CYP3A4 (0.46) KMT2ACYP3A4RARARARBRARG
SCHEMBL6591418 0.67 RARA (0.46) KMT2ACYP3A4RARARARBRARG
SCHEMBL6591282 0.67 MAPT (0.34) KMT2ACYP3A4RARARARBRARG
SCHEMBL8558273 0.66 RARA (0.56) KMT2ACYP3A4RARARARBRARG
SCHEMBL9007075 0.66 RARB (0.49) KMT2ACYP3A4RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958954-A 2,2-DIALKYL-4-ARYL-SUBSTITUTED BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES ALLERGAN SALES, INC. (US) 1999-09-28 US disclosed