SCHEMBL6592969

SCHEMBL6592969

CCOC(=O)c1ccc(C#Cc2cc3c(cc2OC)SC(C)(C)C=C3OS(=O)(=O)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 2/20 0.34
CYP3A4 P08684 1/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
HPGD P15428 2/20 0.33
HSD17B2 P37059 1/20 0.33
LMNA P02545 1/20 0.33
ACHE P22303 1/20 0.33
MAPT P10636 2/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPK1 P28482 1/20 0.32
STS P08842 1/20 0.31
PDK2 Q15119 2/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1140980 0.91 RARA (0.39) NPC1RAB9ASMN1; SMN2KMT2ACYP3A4
SCHEMBL6591282 0.90 MAPT (0.34) KMT2ACYP3A4RARARARBRARG
SCHEMBL6588869 0.82 CYP3A4 (0.53) NPC1RAB9ASMN1; SMN2KMT2ACYP3A4
SCHEMBL6591025 0.81 KMT2A (0.33) NPC1KMT2ACYP3A4RARARARB
SCHEMBL5669671 0.80 RARB (0.41) CYP3A4RARARARBRARG
SCHEMBL6591418 0.79 RARA (0.46) KMT2ACYP3A4RARARARBRARG
SCHEMBL6234971 0.78 PDK2 (0.38) NPC1RAB9ASMN1; SMN2KMT2ACYP3A4
SCHEMBL8333199 0.77 KMT2A (0.35) NPC1RAB9ASMN1; SMN2KMT2ACYP3A4
SCHEMBL6591370 0.76 KMT2A (0.41) NPC1RAB9ASMN1; SMN2KMT2ACYP3A4
SCHEMBL6590616 0.75 CYP3A4 (0.35) NPC1RAB9ASMN1; SMN2KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042313-B1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
EP-1042313-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY Allergan Sales, Inc. (US) 2000-10-11 EP disclosed
US-5958954-A 2,2-DIALKYL-4-ARYL-SUBSTITUTED BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES ALLERGAN SALES, INC. (US) 1999-09-28 US disclosed
WO-1999033821-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST-LIKE ACTIVITY ALLERGAN SALES, INC. (US) 1999-07-08 WO disclosed