SCHEMBL8334176

SCHEMBL8334176

COc1ccc(N(C(=N)N)c2ccc3c4c(cccc24)C=C3)c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
EP300 Q09472 1/20 0.37
KAT8 Q9H7Z6 1/20 0.37
SCN2A Q99250 1/20 0.33
PLAU P00749 2/20 0.33
PLK1 P53350 1/20 0.33
IMPDH2 P12268 1/20 0.33
IMPDH1 P20839 1/20 0.33
CDC25B P30305 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
STAT6 P42226 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HPGDS O60760 1/20 0.32
MAPT P10636 4/20 0.32
TUBB3 Q13509 1/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803077 0.87 IDO1 (0.49) IDO1EP300KAT8PLAUPLK1
SCHEMBL9112765 0.85 SIGMAR1 (0.33) SIGMAR1
SCHEMBL6717206 0.84 SIGMAR1 (0.47) IDO1EP300KAT8PLK1IMPDH2
Hydrochloric Acid SCHEMBL8711879 0.82 SIGMAR1 (0.46) IDO1EP300KAT8PLK1IMPDH2
SCHEMBL9112697 0.82 CHEK1 (0.41) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL6155369 0.81 SIGMAR1 (0.31) SIGMAR1
SCHEMBL6158953 0.80 SIGMAR1 (0.39) SIGMAR1
SCHEMBL6154831 0.78 KDM4E (0.40) IMPDH2IMPDH1ALDH1A1MAPTKDM4E
SCHEMBL9115242 0.76 CTSB (0.40) ALDH1A1CYP3A4HSD17B10MAPTLMNA
SCHEMBL6720796 0.75 SCN2A (0.36) SCN2APLK1CDC25BALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999002145-A1 COMBINATION DRUG THERAPIES COMPRISING AMINOGLYCOSIDE ANTIBIOTICS AND N,N'-DISUBSTITUTED GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1999-01-21 WO disclosed