SCHEMBL8337355

SCHEMBL8337355

O=C(NCc1ccc(C(=O)O)c(C(=O)O)c1)c1cc(-c2ccc(OC(F)(F)F)cc2)cs1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 7/20 0.60
MMP13 P45452 1/20 0.53
MAPK1 P28482 2/20 0.46
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45
PPARA Q07869 4/20 0.45
PPARD Q03181 2/20 0.45
EPHX2 P34913 2/20 0.43
NR1H4 Q96RI1 1/20 0.43
PPARG P37231 1/20 0.43
HTR2C P28335 1/20 0.43
MAPK14 Q16539 1/20 0.43
ABL1 P00519 1/20 0.43
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42
IGF2BP2 Q9Y6M1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6881373 0.92 MMP12 (0.55) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6663858 0.88 MMP12 (0.59) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6462719 0.86 MMP12 (0.64) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6456507 0.85 MMP12 (0.72) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6458023 0.85 MMP12 (0.56) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6874175 0.84 MMP12 (0.57) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6881497 0.83 DHODH (0.48) MMP12
SCHEMBL6450465 0.83 MMP12 (0.62) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6881245 0.83 MMP12 (0.57) MMP12MMP13MAPK1ROCK2ROCK1
SCHEMBL6456642 0.81 MMP12 (0.56) MMP12MMP13MAPK1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018448-A1 NOVEL THIOPHENE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME WARNER-LAMBERT COMPANY LLC (US) 2004-03-04 WO disclosed