SCHEMBL8338455

SCHEMBL8338455

Cc1cccc(-c2c(C(=O)c3ccc(O)cc3)sc3cc(O)ccc23)c1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.66
ESR2 Q92731 2/20 0.48
CNR2 P34972 4/20 0.46
CNR1 P21554 2/20 0.46
MAOB P27338 1/20 0.43
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8341726 0.89 ESR1 (0.74) ESR1ESR2MAOB
SCHEMBL8341280 0.86 ESR1 (0.86) ESR1ESR2MAOB
SCHEMBL8341396 0.86 ESR1 (0.76) ESR1ESR2HSD17B1HSD17B2
SCHEMBL11599689 0.82 ESR1 (0.71) ESR1ESR2
SCHEMBL21260801 0.81 ESR1 (0.78) ESR1ESR2MAOB
SCHEMBL15660907 0.80 ESR1 (1.00) ESR1ESR2MAOB
SCHEMBL11600001 0.79 ESR1 (0.67) ESR1ESR2
SCHEMBL8338171 0.79 ESR1 (0.63) ESR1MAOBHSD17B1HSD17B2
SCHEMBL8337732 0.79 ESR1 (0.77) ESR1ESR2
SCHEMBL8340581 0.77 ESR1 (0.74) ESR1ESR2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908859-A ESPECIALLY HYPERCHOLESTEROLEMIA ELI LILLY AND COMPANY (US) 1999-06-01 US disclosed
EP-0897918-A1 Benzothiophene derivatives and their use as pharmaceutically active agents ELI LILLY AND COMPANY (US) 1999-02-24 EP disclosed