SCHEMBL8338540

SCHEMBL8338540

N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccccc1NC(=O)[C@@H](N)Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.60
HDAC4 P56524 3/20 0.60
HDAC1 Q13547 3/20 0.60
HDAC7 Q8WUI4 3/20 0.60
HDAC2 Q92769 3/20 0.60
HDAC10 Q969S8 3/20 0.60
HDAC11 Q96DB2 3/20 0.60
HDAC8 Q9BY41 3/20 0.60
HDAC6 Q9UBN7 3/20 0.60
HDAC9 Q9UKV0 3/20 0.60
HDAC5 Q9UQL6 3/20 0.60
ALPI P09923 1/20 0.56
PKM P14618 1/20 0.56
PTGS1 P23219 1/20 0.56
XIAP P98170 1/20 0.56
SLC7A5 Q01650 1/20 0.56
SLC15A1 P46059 1/20 0.53
CTSC P53634 1/20 0.52
BACE1 P56817 2/20 0.52
LNPEP Q9UIQ6 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6719263 0.84 POLB (0.63) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL28552924 0.84 SMN1; SMN2 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL30454499 0.84 ATM (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL21880156 0.84 SMN1; SMN2 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28277701 0.84 POLB (0.63) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL28279152 0.84 ROCK2 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3255718 0.82 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2312361 0.81 BACE1 (0.63) HDAC8ALPIPKMPTGS1XIAP
SCHEMBL2312372 0.81 BACE1 (0.63) HDAC8ALPIPKMPTGS1XIAP
SCHEMBL28279157 0.81 BACE1 (0.63) HDAC8ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004101494-A1 CALPAIN INHIBITORS CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (ES) 2004-11-25 WO disclosed