SCHEMBL8339113

SCHEMBL8339113

Cc1cn(-c2ccnc3c(F)cccc23)cc1C(=O)N=C(N)N

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 9/20 0.42
HTR5A P47898 3/20 0.41
BTK Q06187 1/20 0.37
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PIK3R2 O00459 1/20 0.36
SLC9A2 Q9UBY0 3/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
SLC9A3 P48764 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8338997 0.81 HTR5A (0.41) SLC9A1HTR5AKDM4EL3MBTL1
SCHEMBL6082191 0.81 BTK (0.36) BTKKDM4EL3MBTL1PIK3R2PTGDR2
SCHEMBL8346528 0.80 RORC (0.38) SLC9A1HTR5AKDM4EL3MBTL1PIK3R2
SCHEMBL6081996 0.69 PIK3R2 (0.43) KDM4EL3MBTL1PIK3R2
SCHEMBL6082339 0.67 CDK8 (0.36) KDM4EL3MBTL1PIK3R2
SCHEMBL25205591 0.67 PIK3R2 (0.38) KDM4EL3MBTL1PIK3R2
SCHEMBL31095534 0.67 PIK3R2 (0.38) KDM4EL3MBTL1PIK3R2
SCHEMBL6083005 0.67 CD38 (0.41)
SCHEMBL6082100 0.67 ADORA2A (0.36) KDM4EL3MBTL1
SCHEMBL9907824 0.66 HTR5A (0.56) SLC9A1HTR5APTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004007478-A2 DERIVATIVES OF 3-GUANIDINOCARBONYL-1-HETEROARYL-PYRROLE, PROCESS FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL USE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-01-22 WO disclosed