SCHEMBL8340988

SCHEMBL8340988

Cc1ccc2c(c1)CN(C)C=C2

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 10/20 0.36
SLC6A4 P31645 10/20 0.36
SLC6A3 Q01959 10/20 0.36
CYP2D6 P10635 1/20 0.33
SRD5A1 P18405 4/20 0.32
HSD17B10 Q99714 1/20 0.32
NOTUM Q6P988 1/20 0.31
ALDH1A1 P00352 1/20 0.30
METAP1 P53582 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22796908 0.85 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3HSD17B10ALDH1A1
SCHEMBL29809557 0.85 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3HSD17B10ALDH1A1
SCHEMBL23346755 0.79 MAPT (0.34) HSD17B10ALDH1A1
SCHEMBL16654882 0.79 SLC6A4 (0.36) SLC6A2SLC6A4SLC6A3SRD5A1NOTUM
SCHEMBL21933883 0.77 SLC6A2 (0.30) SLC6A2SLC6A4SLC6A3SRD5A1
SCHEMBL14085050 0.77 BRD4 (0.40) SLC6A2SLC6A4SLC6A3SRD5A1ALDH1A1
SCHEMBL30385312 0.74 HDAC3 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6HSD17B10
SCHEMBL1564351 0.74 HDAC3 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6HSD17B10
Hydrochloric Acid SCHEMBL187276 0.72 MAOA (0.41) SLC6A2SLC6A4SLC6A3CYP2D6HSD17B10
Iodide SCHEMBL4322466 0.72 HDAC3 (0.40) SLC6A2SLC6A4SLC6A3CYP2D6HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041842-B1 SPIROCYCLIC COMPOUNDS AS TRYPTOPHAN HYDROXYLASE INHIBITORS KAROS PHARMACEUTICALS INC (US) 2019-10-23 EP disclosed
WO-2004014384-A2 CYCLIC COMPOUNDS CONTAINING ZINC BINDING GROUPS AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed