SCHEMBL8342148

SCHEMBL8342148

CC(=O)c1c(C)oc2c(NC(=O)c3c(Cl)ccc(N)c3Cl)cccc12

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.44
GAA P10253 1/20 0.39
LMNA P02545 3/20 0.38
ALDH1A1 P00352 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TP53 P04637 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CXCR2 P25025 1/20 0.36
PKM P14618 2/20 0.36
NPC1 O15118 1/20 0.36
GPR35 Q9HC97 3/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7827793 0.89 JAK1 (0.45) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL7815986 0.89 MAPT (0.39) MAPTLMNAALDH1A1NPSR1TP53
SCHEMBL7826306 0.87 GAA (0.45) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL7816589 0.87 MAPT (0.44) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL7816264 0.84 TYK2 (0.47) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL7827125 0.83 MAPT (0.43) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL8341717 0.83 GPR35 (0.44) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL7831900 0.81 MAPT (0.40) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL7831814 0.78 RAB9A (0.42) MAPTLMNAALDH1A1NPSR1TP53
SCHEMBL7829562 0.77 MAPT (0.47) MAPTLMNAALDH1A1NPSR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5858995-A ADMINISTERING TO HUMANS AND ANIMALS IN THE TREATMENT OF DISEASES CAUSED BY ABNORMAL BONE METABOLISM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-01-12 US disclosed
EP-0757682-A1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029907-A1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-09 WO disclosed