SCHEMBL8343307

SCHEMBL8343307

CS(=O)(=O)N1c2ccccc2C2(CCNCC2)C1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.50
ICAM1 P05362 2/20 0.50
ITGAL P20701 2/20 0.50
MMP2 P08253 8/20 0.47
MMP9 P14780 8/20 0.47
ALOX15 P16050 1/20 0.47
ACE P12821 3/20 0.47
GHSR Q92847 1/20 0.45
KMT2A Q03164 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8346758 0.91 TACR1 (0.51) MMP2MMP9GHSR
SCHEMBL8346990 0.90 TACR1 (0.53) KMT2AMEN1
SCHEMBL8345542 0.89 TACR1 (0.55)
SCHEMBL8343109 0.89 TACR1 (0.55)
SCHEMBL8345475 0.89 TACR1 (0.42) ITGB2ICAM1ITGALMMP2MMP9
SCHEMBL8346929 0.85 TACR1 (0.56) GHSR
SCHEMBL8349377 0.85 TACR1 (0.48) MMP9GHSR
SCHEMBL7399209 0.84 GHSR (0.47) MMP2MMP9ACEGHSR
SCHEMBL8345132 0.83 TACR1 (0.53) MMP9GHSR
SCHEMBL8344898 0.82 TACR1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869489-A TREATMENT OF INFLAMMATORY DISEASES, MIGRAINES AND ASTHMA MERCK & CO., INC. (US) 1999-02-09 US disclosed