SCHEMBL8346758

SCHEMBL8346758

CS(=O)(=O)N1c2ccccc2C2(CCNCC2)C1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.51
TACR2 P21452 2/20 0.51
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
KCNT1 Q5JUK3 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
HDAC8 Q9BY41 3/20 0.45
HDAC6 Q9UBN7 3/20 0.45
HDAC3 O15379 2/20 0.45
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC10 Q969S8 2/20 0.45
HDAC11 Q96DB2 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8343307 0.91 ITGB2 (0.50) MMP2MMP9GHSR
SCHEMBL8346990 0.89 TACR1 (0.53) TACR1TACR2MAPT
SCHEMBL8343109 0.88 TACR1 (0.55) TACR1TACR2
SCHEMBL8345542 0.88 TACR1 (0.55) TACR1TACR2
SCHEMBL8345475 0.84 TACR1 (0.42) TACR1TACR2MMP2MMP9MMP8
SCHEMBL8346929 0.83 TACR1 (0.56) TACR1TACR2GHSR
SCHEMBL8349377 0.82 TACR1 (0.48) TACR1TACR2MMP9MMP8GHSR
SCHEMBL8344898 0.81 TACR1 (0.52) TACR1TACR2
SCHEMBL8345132 0.81 TACR1 (0.53) TACR1TACR2MMP9MMP8GHSR
SCHEMBL7399209 0.80 GHSR (0.47) MMP2MMP9GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869489-A TREATMENT OF INFLAMMATORY DISEASES, MIGRAINES AND ASTHMA MERCK & CO., INC. (US) 1999-02-09 US disclosed