SCHEMBL8345010

SCHEMBL8345010

Cc1cnc2c(c1)c(=O)n(C)c1nccn21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
KAT2B Q92831 3/20 0.33
HPGD P15428 3/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
PARG Q86W56 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 2/20 0.30
HTT P42858 1/20 0.30
WEE1 P30291 1/20 0.30
BRD4 O60885 1/20 0.30
PDE6A P16499 1/20 0.30
PDE6B P35913 1/20 0.30
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE4D Q08499 1/20 0.30
PDE1C Q14123 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8342935 0.77 GABRA1 (0.38) ALDH1A1KDM4EMAPTHTT
SCHEMBL26602715 0.74
SCHEMBL30625233 0.74
SCHEMBL8345008 0.73 AAK1 (0.35) ALDH1A1HPGDGAAMAPTBRD4
SCHEMBL30625223 0.71 KDM4E (0.33) ALDH1A1L3MBTL1KDM4EHPGDGAA
SCHEMBL26602768 0.71 KDM4E (0.33) ALDH1A1L3MBTL1KDM4EHPGDGAA
SCHEMBL30625103 0.70
SCHEMBL26602577 0.70
SCHEMBL30625252 0.70
SCHEMBL26602737 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014384-A2 CYCLIC COMPOUNDS CONTAINING ZINC BINDING GROUPS AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed