SCHEMBL8345013

SCHEMBL8345013

COC(=O)CC1CCc2ncccc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.38
ALDH1A1 P00352 5/20 0.36
MIF P14174 1/20 0.36
JAK2 O60674 1/20 0.35
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTT P42858 1/20 0.34
PDE10A Q9Y233 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
DGAT1 O75907 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL924605 0.80 HTR1A (0.43) CYP19A1ALDH1A1MIF
SCHEMBL31374633 0.79 ALDH1A1 (0.52) CYP19A1ALDH1A1KDM4ESMN1; SMN2DGAT1
SCHEMBL6644734 0.79 ALDH1A1 (0.52) CYP19A1ALDH1A1KDM4ESMN1; SMN2DGAT1
SCHEMBL923006 0.74 CYP19A1 (0.46) CYP19A1DGAT1
SCHEMBL924439 0.74 CYP19A1 (0.46) CYP19A1ALDH1A1MIFSMN1; SMN2
Bromide SCHEMBL8124970 0.73 CYP19A1 (0.45) CYP19A1DGAT1
SCHEMBL9836578 0.72 HTR2C (0.47) MIFHTTCYP1A2
SCHEMBL2877889 0.72 MAPT (0.47) ALDH1A1KDM4EGAAHPGDNPSR1
SCHEMBL27654667 0.71 GAA (0.38) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL9855381 0.70 CYP26A1 (0.60) CYP19A1ALDH1A1SMN1; SMN2DGAT1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935956-A Pyridazine compounds ASTRA PHARMACEUTICALS LTD. (GB) 1999-08-10 US disclosed