SCHEMBL8345262

SCHEMBL8345262

N#Cc1cccc2c(=O)c3cc(-c4ccccc4)cnc3ccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 7/20 0.51
KCNH2 Q12809 2/20 0.46
ALDH1A1 P00352 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MAPK10 P53779 1/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
GRIN2B Q13224 1/20 0.40
PSMB5 P28074 1/20 0.39
SSTR2 P30874 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910843 0.83 ALDH1A1 (0.55) METKCNH2ALDH1A1TDP1NPSR1
SCHEMBL7144926 0.82 MET (0.43) METCA1CA2EGFR
SCHEMBL2449685 0.80 MET (0.54) METKCNH2MAPK10PSMB5
SCHEMBL2450265 0.80 MET (0.68) METKCNH2MAPK10PSMB5
SCHEMBL2447320 0.80 MET (0.54) METKCNH2ALDH1A1NPSR1MAPK10
SCHEMBL4309790 0.78 MET (0.57) METKCNH2KDM4EMAPK10PSMB5
SCHEMBL2447746 0.77 MET (0.51) METKCNH2MAPK10PSMB5
SCHEMBL2330707 0.76 MET (0.67) METKCNH2MAPK10
SCHEMBL2448087 0.76 MET (0.58) METKCNH2MAPK10PSMB5
SCHEMBL8344609 0.75 MET (0.49) METGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003084931-A1 5H-BENZO[4,5]CYCLOHEPTA[1,2-B]PYRIDINE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2003-10-16 WO disclosed