SCHEMBL83482

SCHEMBL83482

N#Cc1c(F)cc(-c2c(O)cc(O)cc2F)cc1F

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.44
ESR2 Q92731 10/20 0.44
TRPV4 Q9HBA0 1/20 0.42
NQO1 P15559 1/20 0.42
AR P10275 3/20 0.41
EGLN2 Q96KS0 2/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL83963 0.93 NQO1 (0.50) ESR1ESR2TRPV4NQO1AR
SCHEMBL30332317 0.91 ESR1 (0.51) ESR1ESR2TRPV4AREGLN2
SCHEMBL81244 0.82 TRPV4 (0.58) ESR1ESR2TRPV4AREGLN2
SCHEMBL16748052 0.77 ESR1 (0.47) ESR1ESR2TRPV4AR
SCHEMBL16748051 0.77 ESR1 (0.54) ESR1ESR2TRPV4AR
SCHEMBL84047 0.76 NQO1 (0.46) ESR1ESR2NQO1ARCNR2
SCHEMBL12840889 0.73 TRPV4 (0.38) ESR1ESR2TRPV4AREGLN2
SCHEMBL16604331 0.72 TRPV4 (0.47) ESR1ESR2TRPV4EGLN2PDE4A
SCHEMBL8063680 0.72 ESR1 (0.53) ESR1ESR2TRPV4AR
SCHEMBL16922703 0.70 TRPV4 (0.45) ESR1ESR2TRPV4EGLN2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129002-B2 Compounds for use in liquid crystal media MERCK PATENT GMBH (DE) 2012-03-06 US disclosed
US-7419706-B2 Liquid crystalline medium MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2008-09-02 US disclosed