SCHEMBL8348223

SCHEMBL8348223

Fc1ccccc1-c1nccc(Nc2ccncc2)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 10/20 0.59
CYP3A4 P08684 10/20 0.59
CYP2D6 P10635 7/20 0.59
CYP2C19 P33261 7/20 0.59
ALDH1A1 P00352 5/20 0.59
USP2 O75604 3/20 0.58
TSHR P16473 1/20 0.58
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
BUB1 O43683 2/20 0.53
AURKA O14965 3/20 0.46
TGFBR1 P36897 1/20 0.44
MAPK1 P28482 4/20 0.44
NPC1 O15118 2/20 0.44
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
CHEK1 O14757 1/20 0.44
IKBKB O14920 1/20 0.44
PDPK1 O15530 1/20 0.44
CHEK2 O96017 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8344338 0.89 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8345893 0.84 CYP1A2 (0.48) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8347442 0.84 BUB1 (0.51) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8348278 0.83 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8345329 0.82 TGFBR1 (0.58) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8346049 0.78 ABCG2 (0.67) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL16392231 0.76 ABCB1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8345669 0.75 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL18114578 0.75 KDR (0.60) MAPK1CHEK1PDPK1CHEK2PRKCG
SCHEMBL28296096 0.72 NPC1 (0.50) CYP1A2CYP3A4TSHRKMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004024159-A1 INHIBITORS OF TFGβ SCIOS INC. (US) 2004-03-25 WO disclosed