SCHEMBL8348277

SCHEMBL8348277

COC(=O)c1cc(N)ccc1-c1ncco1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 4/20 0.58
GAA P10253 3/20 0.47
GLRA3 O75311 1/20 0.44
GLRB P48167 1/20 0.44
CYP46A1 Q9Y6A2 1/20 0.41
ABCB1 P08183 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
GLA P06280 2/20 0.39
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TUBB4A P04350 3/20 0.38
TUBB P07437 3/20 0.38
TUBA3C P0DPH7 3/20 0.38
TUBA1B P68363 3/20 0.38
TUBA4A P68366 3/20 0.38
TUBB4B P68371 3/20 0.38
TUBB3 Q13509 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16463175 0.85 CYP46A1 (0.58) CFTRGLRA3GLRBCYP46A1ALDH1A1
SCHEMBL16114117 0.84 CFTR (0.55) CFTRGLRA3GLRBCYP46A1TUBB4A
SCHEMBL29469507 0.84 CFTR (0.52) CFTRGAAGLRA3GLRBCYP46A1
SCHEMBL305696 0.80 CFTR (0.53) CFTRGLRA3GLRBALDH1A1KDM4E
SCHEMBL8347921 0.80 CFTR (0.48) CFTRGLRA3GLRBCYP46A1ALDH1A1
SCHEMBL9705197 0.79 GAA (0.65) CFTRGAACYP46A1ABCB1ALDH1A1
SCHEMBL8347738 0.78 CFTR (0.47) CFTRGLRA3GLRBCYP46A1KDM4E
SCHEMBL2726214 0.75 CFTR (0.58) CFTRGAAABCB1ALDH1A1KDM4E
SCHEMBL29469477 0.75 ALDH1A1 (0.51) CFTRGAAGLRA3GLRBCYP46A1
SCHEMBL16197237 0.73 GAA (0.47) CFTRGAACYP46A1ABCB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004000788-A1 UREIDO-SUBSTITUTED ANILINE COMPOUNDS USEFUL AS SERINE PROTEASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-31 WO disclosed