SCHEMBL8348292

SCHEMBL8348292

COCCOCN(c1onc(C)c1C)S(=O)(=O)c1ccccc1-c1ncccn1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 10/20 0.48
EDNRB P24530 5/20 0.41
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8568832 0.93 EDNRA (0.52) EDNRAEDNRB
SCHEMBL8351866 0.90 EDNRA (0.50) EDNRAEDNRBTP53MAPT
SCHEMBL8568463 0.87 EDNRA (0.53) EDNRAEDNRB
SCHEMBL6772184 0.86 EDNRA (0.38) EDNRAEDNRBTP53MAPT
SCHEMBL6640800 0.86 EDNRB (0.41) EDNRAEDNRBTP53MAPT
SCHEMBL8685211 0.86 EDNRA (0.41) EDNRAEDNRB
SCHEMBL8687989 0.86 EDNRA (0.40) EDNRAEDNRBTP53MAPT
SCHEMBL9089818 0.85 EDNRA (0.37) EDNRAEDNRBTP53MAPT
SCHEMBL8353066 0.85 EDNRA (0.51) EDNRAEDNRBTP53MAPT
SCHEMBL6961532 0.85 EDNRA (0.54) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939446-A HYPOTENSIVE AGENTS FROM ISOXAZOLESULFONAMIDES BRISTOL-MYERS SQUIBB CO. (US) 1999-08-17 US disclosed