SCHEMBL8348494

SCHEMBL8348494

CCC(C1(c2ccc(Cl)c(Cl)c2)CCN(C(=O)c2ccc(OC)cc2)C1)S(=O)(=O)O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 3/20 0.50
TACR1 P25103 3/20 0.50
HTR1A P08908 1/20 0.44
CYP1A2 P05177 3/20 0.43
USP2 O75604 2/20 0.43
HIF1A Q16665 1/20 0.43
TSHR P16473 4/20 0.43
CYP2D6 P10635 4/20 0.42
MAPK1 P28482 1/20 0.42
CYP3A4 P08684 4/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8349962 0.93 TACR2 (0.50) TACR2TACR1TSHRALDH1A1
SCHEMBL8355974 0.91 CA12 (0.42) TACR2TACR1CYP2D6CYP3A4KMT2A
SCHEMBL8355522 0.90 TACR2 (0.53) TACR2TACR1HTR1AALDH1A1
SCHEMBL8347396 0.89 TACR2 (0.48) TACR2TACR1CYP2D6CYP3A4
SCHEMBL8350232 0.88 TACR2 (0.52) TACR2TACR1TSHRKMT2AALDH1A1
SCHEMBL8347206 0.88 TACR2 (0.51) TACR2TACR1
SCHEMBL8356065 0.87 KMT2A (0.39) TACR2TACR1MEN1KMT2AALDH1A1
SCHEMBL8350410 0.85 KMT2A (0.38) TACR2TACR1KMT2A
SCHEMBL8355501 0.85 TACR2 (0.51) TACR2TACR1MEN1KMT2A
SCHEMBL8350132 0.84 TACR2 (0.53) TACR2TACR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861416-A TREATMENT OF ASTHMA OR COUGH MERRELL PHARMACEUTICALS INC. (US) 1999-01-19 US disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed