SCHEMBL8349971

SCHEMBL8349971

CCc1c(C)nc2ccc(Br)cc2c1C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.66
HTT P42858 2/20 0.66
RXFP1 Q9HBX9 5/20 0.63
CYP1A2 P05177 2/20 0.63
CYP2C9 P11712 2/20 0.63
CYP2C19 P33261 2/20 0.63
CYP2D6 P10635 1/20 0.63
AURKA O14965 2/20 0.60
AURKB Q96GD4 2/20 0.60
KDR P35968 1/20 0.60
PRNP P04156 3/20 0.58
PPARG P37231 2/20 0.58
NR2E3 Q9Y5X4 2/20 0.58
NCOR2 Q9Y618 2/20 0.58
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
TP53 P04637 1/20 0.56
DHODH Q02127 3/20 0.52
LMNA P02545 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13136430 0.84 ALDH1A1 (0.60) ALDH1A1HTTRXFP1CYP1A2CYP2C9
SCHEMBL17593966 0.83 DHODH (0.71) ALDH1A1HTTRXFP1AURKAAURKB
SCHEMBL1305487 0.83 ALDH1A1 (0.85) ALDH1A1HTTRXFP1CYP1A2CYP2C9
SCHEMBL28225220 0.82 ALDH1A1 (0.57) ALDH1A1HTTRXFP1CYP1A2CYP2C9
SCHEMBL15486910 0.81 ALDH1A1 (0.71) ALDH1A1HTTRXFP1CYP1A2CYP2C9
SCHEMBL14595374 0.79 PDE10A (0.66) HTTRXFP1MEN1KMT2ASMN1; SMN2
SCHEMBL15487148 0.77 DHODH (0.56) ALDH1A1HTTRXFP1CYP1A2CYP2C9
SCHEMBL31271707 0.76 ALDH1A1 (0.64) ALDH1A1HTTRXFP1AURKAAURKB
SCHEMBL17593896 0.76 PTGFR (0.65) RXFP1AURKAAURKBKDRPRNP
SCHEMBL15486934 0.75 ALDH1A1 (0.56) ALDH1A1HTTRXFP1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629468-B2 Neuroprotectants, analgesics or anticonvulsants JANSSEN PHARMACEUTICA NV (BE) 2009-12-08 US disclosed
US-7629468-B2 Neuroprotectants, analgesics or anticonvulsants JANSSEN PHARMACEUTICA NV (BE) 2009-12-08 US disclosed
US-7517517-B2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-14 US disclosed
US-7517517-B2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-14 US disclosed
WO-2003082350-A2 RADIOLABELLED QUINOLINE AND QUINOLINONE DERIVATIVES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR LIGANDS JANSSEN PHARMACEUTICA N.V. (BE) 2003-10-09 WO disclosed