SCHEMBL8350133

SCHEMBL8350133

Fc1ccccc1C#Cc1ccc(COCl)o1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.35
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
PRSS3 P35030 1/20 0.33
GRM5 P41594 2/20 0.33
EGFR P00533 1/20 0.31
ERBB2 P04626 1/20 0.31
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL256077 0.80 GRM5 (0.38) PTGDR2PRSS1PRSS2PRSS3GRM5
SCHEMBL2109413 0.71 GRM5 (0.39) PTGDR2PRSS1PRSS2PRSS3GRM5
SCHEMBL9967683 0.69 GRM5 (0.39) PTGDR2PRSS1PRSS2PRSS3GRM5
SCHEMBL6805955 0.69 PRSS1 (0.44) PTGDR2PRSS1PRSS2PRSS3GRM5
SCHEMBL29251289 0.69 GRM5 (0.52) PTGDR2GRM5ALDH1A1SMN1; SMN2
SCHEMBL2109417 0.68 ALDH1A1 (0.37) PTGDR2PRSS1PRSS2PRSS3GRM5
SCHEMBL8278416 0.67 PRSS1 (0.45) PTGDR2PRSS1PRSS2PRSS3GRM5
Fluoride SCHEMBL31286347 0.67 GRM5 (0.50) PTGDR2GRM5ALDH1A1SMN1; SMN2
Charcoal, Activated SCHEMBL31286314 0.67 GRM5 (0.50) PTGDR2GRM5ALDH1A1SMN1; SMN2
SCHEMBL6810736 0.66 ALDH1A1 (0.48) PTGDR2PRSS1PRSS2PRSS3GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060884-A1 [4-(3-AMINOMETHYLPHENYL) PIPERIDIN-1-YL]- [5-(2-FLUOROPHENYLETHYNYL)FURAN-2-YL]-METHANONE AS AN INHIBITOR OF MAST CELL TRYPTASE AVENTIS PHARMACEUTICALS INC. (US) 2004-07-22 WO disclosed