SCHEMBL8352129

SCHEMBL8352129

CCN1CCN(c2cccc(CC(C)(C)C)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.56
DRD2 P14416 7/20 0.49
GAA P10253 2/20 0.49
RAD52 P43351 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MAPT P10636 1/20 0.49
GFER P55789 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KHK P50053 2/20 0.46
SIGMAR1 Q99720 1/20 0.45
DRD3 P35462 2/20 0.44
AGXT P21549 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4577137 0.85 CHRNA7 (0.49) CHRNA7DRD2GAARAD52KDM4E
SCHEMBL4577142 0.85 CHRNA7 (0.49) CHRNA7DRD2GAARAD52KDM4E
SCHEMBL10190899 0.84 AGXT (0.61) DRD2GAAKDM4EMAPTGFER
SCHEMBL8349954 0.84 PRMT6 (0.59) GAAKDM4EMAPTAGXT
SCHEMBL10190904 0.83 PRMT6 (0.62) GAAKDM4EMAPTAGXT
SCHEMBL8352403 0.83 DRD2 (0.50) DRD2SIGMAR1DRD3AGXT
SCHEMBL8348977 0.82 DRD2 (0.52) DRD2MAPTSIGMAR1AGXT
SCHEMBL2376462 0.81 CHRNA7 (0.59) CHRNA7DRD2GAARAD52KDM4E
SCHEMBL8349952 0.81 KHK (0.45) KDM4EMAPTSMN1; SMN2KHKAGXT
SCHEMBL20671914 0.80 ADRB1 (0.57) DRD2MAPTSIGMAR1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003020278-A1 CYSTEINE PROTEASE INHIBITORS WITH 2-CYANO-4-AMINO-PYRIMIDINE STRUCTURE AND CATHEPSIN K INHIBITORY ACTIVITY FOR THE TREATMENT OF INFLAMMATIONS AND OTHER DISEASES NOVARTIS AG (CH) 2003-03-13 WO disclosed