SCHEMBL8352575

SCHEMBL8352575

Cc1cc([S+](N)[O-])c(C=C2c3ccccc3CCc3ccccc32)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34
AR P10275 1/20 0.34
CYP3A4 P08684 4/20 0.33
CYP1A2 P05177 3/20 0.33
RET P07949 3/20 0.33
CYP2C19 P33261 2/20 0.33
MAPT P10636 5/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
KMT2A Q03164 3/20 0.33
PKM P14618 1/20 0.33
STAT3 P40763 1/20 0.33
STAT1 P42224 1/20 0.33
CYP2D6 P10635 3/20 0.32
SLC6A2 P23975 4/20 0.32
TP53 P04637 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4168482 0.77 NR3C1 (0.42) NR3C1PGRNR3C2ARMAPT
SCHEMBL4163483 0.74 NR3C1 (0.42) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL4163517 0.71 TSHR (0.40) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL4160618 0.69 MAPT (0.56) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL4167052 0.68 NPC1 (0.46) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL4167049 0.68 NPC1 (0.46) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL4161295 0.68 KMT2A (0.44) ALDH1A1SMN1; SMN2KMT2ALMNAMEN1
SCHEMBL4175519 0.68 NR3C1 (0.39) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL8352573 0.67 RAB9A (0.38) NR3C1PGRNR3C2ARCYP3A4
SCHEMBL4157508 0.64 NR3C1 (0.49) NR3C1PGRNR3C2ARCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052847-A2 TRICYCLIC STEROID HORMONE NUCLEAR RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2004-06-24 WO disclosed