SCHEMBL8353620

SCHEMBL8353620

O=C1NC(=O)c2c1c1c3cc(O)ccc3[nH]c1c1c2c2ccccc2n1C1C[C@H](O)[C@@H](O)[C@H]1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 3/20 0.56
ROCK2 O75116 7/20 0.55
GSK3A P49840 1/20 0.54
GSK3B P49841 1/20 0.54
CDK5 Q00535 1/20 0.54
CDK5R1 Q15078 1/20 0.54
PRKCQ Q04759 3/20 0.53
CHEK1 O14757 5/20 0.50
WEE1 P30291 4/20 0.50
SRC P12931 1/20 0.50
PRKCA P17252 2/20 0.49
CDK4 P11802 2/20 0.48
CCND1 P24385 2/20 0.48
CCNE2 O96020 1/20 0.46
PRKACA P17612 1/20 0.46
PRKACG P22612 1/20 0.46
PRKACB P22694 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
PRKD3 O94806 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14440450 1.00 TOP1 (0.56) TOP1ROCK2GSK3AGSK3BCDK5
SCHEMBL14440418 0.94 TOP1 (0.63) TOP1ROCK2GSK3AGSK3BCDK5
SCHEMBL14440376 0.93 TOP1 (0.56) TOP1ROCK2GSK3AGSK3BCDK5
SCHEMBL8354746 0.91 CDK4 (0.55) TOP1ROCK2CDK5CDK5R1PRKCQ
SCHEMBL8350893 0.91 PRKCQ (0.63) ROCK2CDK5CDK5R1PRKCQCHEK1
SCHEMBL8352405 0.91 PRKCQ (0.63) ROCK2CDK5CDK5R1PRKCQCHEK1
SCHEMBL14440392 0.90 PRKCQ (0.62) ROCK2CDK5CDK5R1PRKCQCHEK1
SCHEMBL8352230 0.90 PRKCQ (0.62) ROCK2CDK5CDK5R1PRKCQCHEK1
SCHEMBL8355911 0.88 ROCK2 (0.56) TOP1ROCK2PRKCQPRKCACDK4
SCHEMBL14440448 0.88 ROCK2 (0.56) TOP1ROCK2PRKCQPRKCACDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003051887-A1 N-CARBACYCLE MONOSUBSTITUTED INDOLOCARBAZOLES AS PROTEIN KINASE INHIBITORS NAD AG (DE) 2003-06-26 WO disclosed