SCHEMBL8355392

SCHEMBL8355392

Cc1c(F)c(F)c(F)c(C(=O)CBr)c1F

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 14/20 0.42
TAS1R1 Q7RTX1 13/20 0.42
TAS1R2 Q8TE23 13/20 0.42
PTPN1 P18031 1/20 0.36
GSK3B P49841 1/20 0.36
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTT P42858 1/20 0.32
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RECQL P46063 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1481978 0.87 PTPN1 (0.44) PTPN1GSK3BPKMSMN1; SMN2HTT
SCHEMBL22795572 0.76 TAS1R3 (0.46) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2
SCHEMBL13125484 0.73 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2SMN1; SMN2ALDH1A1
SCHEMBL9748198 0.73 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2
SCHEMBL2860749 0.73 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2
SCHEMBL12140043 0.72 TAS1R3 (0.47) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2
SCHEMBL7652879 0.71 TAS1R3 (0.42) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2
SCHEMBL2470702 0.70 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL12629274 0.69 TAS1R3 (0.48) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2
Bicarbonate SCHEMBL27999118 0.69 TAS1R3 (0.41) TAS1R3TAS1R1TAS1R2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877193-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1999-03-02 US disclosed