SCHEMBL7652879

SCHEMBL7652879

Cc1c(F)c(F)c(F)c(C(=O)Cl)c1F

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 14/20 0.42
TAS1R1 Q7RTX1 13/20 0.42
TAS1R2 Q8TE23 13/20 0.42
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HTT P42858 2/20 0.32
KDM4C Q9H3R0 1/20 0.32
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6740803 0.95 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2CES2CES1
SCHEMBL10587923 0.88 TAS1R3 (0.35) TAS1R3TAS1R1TAS1R2CES2CES1
SCHEMBL2777861 0.88 TAS1R3 (0.39) TAS1R3TAS1R1TAS1R2CES2CES1
SCHEMBL1657 0.84 CES2 (0.48) CES2CES1HTTKDM4CPKM
SCHEMBL18774737 0.82 TAS1R3 (0.33) TAS1R3TAS1R1TAS1R2CES2CES1
SCHEMBL9019898 0.82 TAS1R3 (0.40) TAS1R3TAS1R1TAS1R2CES2CES1
SCHEMBL6538271 0.82 CES2 (0.46) CES2CES1HTTPKMSMN1; SMN2
SCHEMBL996758 0.82 CES2 (0.43) CES2CES1HTTPKMSMN1; SMN2
SCHEMBL19307720 0.79 CES2 (0.48) CES2CES1HTTKDM4CPKM
SCHEMBL2860749 0.78 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2PKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380396-B1 CHEMICAL INTERMEDIATES FOR ANTIINFLAMMATORY AGENTS PFIZER INC. 2002-04-30 US disclosed
US-6207678-B1 USED FOR TREATING INFLAMMATORY DISEASE SUCH AS ARTHRITIS, PSORIASIS, ASTHMA OR INFLAMMATORY BOWEL DISEASE, CENTRAL NERVOUS SYSTEM DISORDER SUCH AS ANXIETY, DEPRESSION, DEMENTIA OR PSYCHOSIS, GASTROINTESTINAL DISORDERS PFIZER INC 2001-03-27 US disclosed