SCHEMBL8355604

SCHEMBL8355604

N[C@@H](Cc1ccccc1)C(=O)ON[C@@H](Cc1ccc(O)cc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.55
MME P08473 1/20 0.50
ALPI P09923 1/20 0.50
PKM P14618 1/20 0.50
PTGS1 P23219 1/20 0.50
XIAP P98170 1/20 0.50
ACE P12821 3/20 0.47
OPRD1 P41143 5/20 0.47
OPRM1 P35372 4/20 0.47
OPRK1 P41145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5163110 0.82 ITGA4 (0.43) SLC7A5MMEACEOPRD1OPRM1
SCHEMBL7227998 0.81 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine Methyl Ester SCHEMBL28118728 0.80 SLC7A5 (0.50) SLC7A5MMEOPRD1OPRM1OPRK1
SCHEMBL1422055 0.80 SLC7A5 (0.64) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanyltyrosine SCHEMBL3037096 0.80 MME (0.67) SLC7A5MMEACEOPRD1OPRM1
Phenylalanyltyrosine SCHEMBL31255162 0.80 MME (0.67) SLC7A5MMEACEOPRD1OPRM1
Phenylalanyltyrosine SCHEMBL29803603 0.80 MME (0.67) SLC7A5MMEACEOPRD1OPRM1
Phenylalanyltyrosine SCHEMBL4282059 0.80 MME (0.67) SLC7A5MMEACEOPRD1OPRM1
SCHEMBL8695556 0.80 MME (0.67) SLC7A5MMEACEOPRD1OPRM1
SCHEMBL29531478 0.80 MME (0.67) SLC7A5MMEACEOPRD1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10323062-B2 Pharmaceutical composition for the prevention and treatment of cardiovascular disease comprising the peptide having the ability to inhibit angiotensin-1 converting enzyme as an active ingredient UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2019-06-18 US disclosed
US-10308681-B2 Pharmaceutical composition for the prevention and treatment of cardiovascular disease comprising the peptide having the ability to inhibit angiotensin-1 converting enzyme as an active ingredient UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2019-06-04 US disclosed
US-20180170961-A1 PHARMACEUTICAL COMPOSITION FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE COMPRISING THE PEPTIDE HAVING THE ABILITY TO INHIBIT ANGIOTENSIN-1 CONVERTING ENZYME AS AN ACTIVE INGREDIENT UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2018-06-21 US disclosed
US-20150175654-A1 PHARMACEUTICAL COMPOSITION FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE COMPRISING THE PEPTIDE HAVING THE ABILITY TO INHIBIT ANGIOTENSIN-1 CONVERTING ENZYME AS AN ACTIVE INGREDIENT UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2015-06-25 US disclosed
US-5922839-A SUPPRESSING FORMATION OF ANGIOTENSIN II IN MAMMALS BY ADMINISTERING MIXTURE OF DRIED STOMACH MUCOSA AND ACIDIFYING AGENT TO PRODUCE IN SITU PEPSIN-INHIBITOR PEPTIDE OF 29 AMINO ACIDS AND MOLECULAR WEIGHT OF 3242 DALTONS STEINER ZOLTAN W (DE) 1999-07-13 US disclosed
US-5688762-A Method of treating hypertension using animal stomach mucosa extract and endogenous protease-inhibitor peptides STEINER ZOLTAN W (DE) 1997-11-18 US disclosed