SCHEMBL8358140

SCHEMBL8358140

Clc1ccc(Cc2nc3ccc(OCCCCBr)cc3s2)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
CSNK1D P48730 2/20 0.43
CYP2D6 P10635 2/20 0.41
AURKB Q96GD4 4/20 0.41
CA2 P00918 2/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.38
ALOX5 P09917 1/20 0.38
EPHX2 P34913 1/20 0.38
ALOX5AP P20292 1/20 0.37
CA1 P00915 1/20 0.37
CA4 P22748 1/20 0.37
CYP3A4 P08684 2/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359722 0.99 KMT2A (0.44) KMT2ACSNK1DCYP2D6AURKBCA2
SCHEMBL8355815 0.93 KMT2A (0.47) KMT2ACSNK1DCYP2D6AURKBCA2
Hydrochloric Acid SCHEMBL8357902 0.86 CYP1A2 (0.54) KMT2ACSNK1DCYP2D6AURKBLMNA
SCHEMBL8356250 0.86 CA2 (0.52) KMT2ACSNK1DCYP2D6AURKBCA2
SCHEMBL8361482 0.84 LMNA (0.54) KMT2ACSNK1DCYP2D6AURKBLMNA
SCHEMBL8358021 0.83 HTT (0.44) KMT2AALOX5EPHX2ALDH1A1
SCHEMBL8356218 0.83 LMNA (0.60) KMT2ACSNK1DCYP2D6AURKBLMNA
SCHEMBL8357709 0.83 KMT2A (0.67) KMT2ACSNK1DCYP2D6CA2LMNA
SCHEMBL8361619 0.81 AURKB (0.46) KMT2ACSNK1DCYP2D6AURKBCA2
SCHEMBL8357941 0.81 MAPT (0.48) KMT2ACYP2D6AURKBCA2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919807-A ANTICHOLESTEROL AGENTS DR. KARL THOMAE GMBH (DE) 1999-07-06 US disclosed
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed