SCHEMBL8358348

SCHEMBL8358348

CCCn1c(C2CCCC2)nc2c(=O)[nH]c(=O)[nH]c21

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.46
ADORA2B P29275 6/20 0.45
ADORA2A P29274 5/20 0.45
MEN1 O00255 1/20 0.44
GMNN O75496 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
TSHR P16473 1/20 0.44
PMP22 Q01453 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9170314 0.72 ADORA1 (0.47) ADORA1ADORA2BADORA2AMEN1GMNN
SCHEMBL8578047 0.72 ADORA1 (0.47) ADORA1ADORA2BADORA2AMEN1GMNN
SCHEMBL8355410 0.72 KMT2A (0.60) ADORA1ADORA2BADORA2AMEN1LMNA
SCHEMBL8358874 0.71 KMT2A (0.59) ADORA1ADORA2BADORA2AMEN1LMNA
SCHEMBL1869547 0.69 ADORA2B (0.46) ADORA1ADORA2BADORA2AMEN1GMNN
1,3-Dipropyl-8-Cyclopentylxanthine [Dpcpx] SCHEMBL12648692 0.68 ADORA1 (0.67) ADORA1ADORA2BADORA2AMEN1GMNN
SCHEMBL7617171 0.68 CYP1A2 (0.43) ADORA2AMEN1LMNACYP1A2TSHR
SCHEMBL9173396 0.67 ADORA1 (0.56) ADORA1ADORA2BADORA2AMEN1GMNN
SCHEMBL7618343 0.67 PNP (0.56) ADORA2AMEN1LMNAKMT2A
SCHEMBL7621514 0.67 MEN1 (0.49) ADORA1MEN1LMNATSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031101-A1 ADENOSINE RECEPTOR ANTAGONISTS WITH IMPROVED BIOACTIVITY UNIVERSITY OF SOUTH FLORIDA (US) 1999-06-24 WO disclosed