SCHEMBL8355410

SCHEMBL8355410

CCCn1c(C2CCCC2)nc2c(=O)[nH]c(=O)n(Cc3ccccc3)c21

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.60
ADORA3 P0DMS8 3/20 0.54
ADORA1 P30542 2/20 0.47
ADORA2B P29275 3/20 0.47
ADORA2A P29274 2/20 0.47
MEN1 O00255 7/20 0.46
POLB P06746 1/20 0.46
RAB9A P51151 1/20 0.46
ALDH1A1 P00352 4/20 0.45
NPSR1 Q6W5P4 3/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
KDM4E B2RXH2 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
TPH1 P17752 2/20 0.43
TPH2 Q8IWU9 2/20 0.43
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8358874 0.97 KMT2A (0.59) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL9168640 0.84 KMT2A (0.74) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL8578047 0.83 ADORA1 (0.47) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL9170314 0.80 ADORA1 (0.47) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL8579759 0.80 KMT2A (0.56) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL6154374 0.78 ADORA2B (0.43) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL8577929 0.73 KMT2A (0.70) KMT2AMEN1POLBRAB9AALDH1A1
SCHEMBL8606081 0.72 KMT2A (0.66) KMT2AADORA3MEN1POLBRAB9A
SCHEMBL8358348 0.72 ADORA1 (0.46) KMT2AADORA3ADORA1ADORA2BADORA2A
SCHEMBL8577877 0.72 ADORA2B (0.60) KMT2AADORA3ADORA1ADORA2BADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031101-A1 ADENOSINE RECEPTOR ANTAGONISTS WITH IMPROVED BIOACTIVITY UNIVERSITY OF SOUTH FLORIDA (US) 1999-06-24 WO disclosed