SCHEMBL8359237

SCHEMBL8359237

CCc1cc2c(C)cc(=O)oc2cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 1.00
ALDH1A1 P00352 9/20 0.72
HPGD P15428 8/20 0.72
KDM4E B2RXH2 8/20 0.72
HSD17B10 Q99714 7/20 0.72
AKR1B1 P15121 2/20 0.72
CYP3A4 P08684 1/20 0.72
THRB P10828 1/20 0.72
CASP1 P29466 6/20 0.63
CASP7 P55210 6/20 0.63
CYP1A2 P05177 2/20 0.63
CYP2C19 P33261 1/20 0.63
HTT P42858 1/20 0.60
NCOA3 Q9Y6Q9 1/20 0.60
GLA P06280 4/20 0.57
GAA P10253 4/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
POLB P06746 2/20 0.57
MAPT P10636 2/20 0.56
TSHR P16473 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11442137 0.84 MCL1 (0.72) MCL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL28061597 0.84 MCL1 (0.72) MCL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL8402004 0.84 MCL1 (0.72) MCL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL8359452 0.84 MCL1 (0.72) MCL1ALDH1A1HPGDKDM4EHSD17B10
4-Methylesculetin SCHEMBL29361762 0.84 MCL1 (1.00) MCL1ALDH1A1HPGDKDM4EHSD17B10
4-Methylesculetin SCHEMBL409482 0.84 MCL1 (1.00) MCL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL8593868 0.83 MCL1 (0.71) MCL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL24865598 0.82 ALDH1A1 (0.82) MCL1ALDH1A1HPGDKDM4EHSD17B10
4-Methylesculetin SCHEMBL6839210 0.82 MCL1 (0.96) MCL1ALDH1A1HPGDKDM4EHSD17B10
4-Methylesculetin SCHEMBL27453331 0.82 ALDH1A1 (0.96) MCL1ALDH1A1HPGDKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968940-A CONTAINING A PURINE DERIVATIVE; ANTICARCINOGENIC AGENTS INSTITUTE OF MATERIA MEDICA (CN) 1999-10-19 US disclosed
CN-1187193-A Retinoids and method of use of same INST MATERIA MEDICA (CN) 1998-07-08 CN disclosed
EP-0850233-A1 RETINOIDS AND METHODS OF USE OF SAME THE INSTITUTE OF MATERIA MEDICA OF CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 1998-07-01 EP disclosed
US-5716982-A COUMARIN COMPOUNDS INSTITUTE OF MATERIA MEDICA, AN INSTITUTE OF THE CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 1998-02-10 US disclosed
WO-1996040669-A1 RETINOIDS AND METHODS OF USE OF SAME INSTITUTE OF MATERIA MEDICA, an Institute of the C (CN) 1996-12-19 WO disclosed