SCHEMBL8359246

SCHEMBL8359246

O=C(Cc1ccccc1)N1CCc2c([nH]c(=O)c3ccccc23)C1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.68
HDAC6 Q9UBN7 3/20 0.59
TRPV1 Q8NER1 2/20 0.56
GPX4 P36969 1/20 0.55
PTGDR2 Q9Y5Y4 1/20 0.50
ROCK2 O75116 1/20 0.49
HDAC1 Q13547 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8360509 0.88 PARP1 (0.69) PARP1HDAC6TRPV1GPX4HDAC1
SCHEMBL20817603 0.86 HDAC6 (0.76) HDAC6TRPV1GPX4HDAC1
SCHEMBL8360520 0.85 PARP1 (0.71) PARP1HDAC6TRPV1GPX4HDAC1
SCHEMBL30023116 0.84 PARP1 (0.66) PARP1TRPV1GPX4
SCHEMBL5367984 0.84 PARP1 (0.66) PARP1TRPV1GPX4
SCHEMBL8363111 0.84 PARP1 (0.77) PARP1TRPV1GPX4
SCHEMBL8360521 0.84 PARP1 (0.73) PARP1HDAC6TRPV1GPX4HDAC1
SCHEMBL8360513 0.82 PARP1 (0.77) PARP1TRPV1GPX4
SCHEMBL8363099 0.82 PARP1 (0.67) PARP1HDAC6TRPV1GPX4HDAC1
SCHEMBL8363098 0.81 PARP1 (1.00) PARP1GPX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed