SCHEMBL8359249

SCHEMBL8359249

CN(C)CCN(C)CCC(=O)N1CCc2[nH]c(=O)c3cc(F)ccc3c2C1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.66
ALDH1A1 P00352 5/20 0.51
GAA P10253 2/20 0.51
BAZ2B Q9UIF8 1/20 0.48
MEN1 O00255 2/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359241 0.94 PARP1 (0.71) PARP1ALDH1A1GAABAZ2BMEN1
SCHEMBL8362887 0.87 PARP1 (0.63) PARP1ALDH1A1GAABAZ2BMEN1
SCHEMBL14444052 0.86 PARP1 (0.76) PARP1ALDH1A1GAABAZ2BMEN1
SCHEMBL8359419 0.83 PARP1 (0.74) PARP1ALDH1A1GAABAZ2BMEN1
SCHEMBL8362888 0.82 PARP1 (0.66) PARP1ALDH1A1BAZ2BMEN1MAPT
SCHEMBL8363083 0.82 PARP1 (0.62) PARP1ALDH1A1GAABAZ2BMEN1
SCHEMBL8359236 0.80 PARP1 (1.00) PARP1ALDH1A1GAABAZ2B
SCHEMBL8362892 0.79 PARP1 (0.66) PARP1ALDH1A1BAZ2BMEN1MAPT
SCHEMBL8363075 0.78 PARP1 (0.61) PARP1ALDH1A1GAABAZ2BMEN1
SCHEMBL8362894 0.78 PARP1 (0.70) PARP1ALDH1A1BAZ2BMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed