SCHEMBL8359236

SCHEMBL8359236

O=C(CCN1CCCCC1)N1CCc2[nH]c(=O)c3cc(F)ccc3c2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 1.00
BAZ2B Q9UIF8 1/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
KDR P35968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359238 0.90 PARP1 (1.00) PARP1BAZ2BALDH1A1GAAKDR
SCHEMBL14444052 0.86 PARP1 (0.76) PARP1BAZ2BALDH1A1GAA
SCHEMBL8362901 0.86 PARP1 (1.00) PARP1NPC1ALDH1A1GAA
SCHEMBL8359243 0.86 PARP1 (0.75) PARP1BAZ2BALDH1A1GAA
SCHEMBL8359419 0.85 PARP1 (0.74) PARP1BAZ2BALDH1A1GAA
SCHEMBL8359241 0.83 PARP1 (0.71) PARP1BAZ2BALDH1A1GAA
SCHEMBL30029262 0.82 PARP1 (0.70) PARP1
SCHEMBL8359463 0.81 PARP1 (1.00) PARP1NPC1ALDH1A1
SCHEMBL8359249 0.80 PARP1 (0.66) PARP1BAZ2BALDH1A1GAA
SCHEMBL8362899 0.78 PARP1 (0.84) PARP1BAZ2BALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed