SCHEMBL8359284

SCHEMBL8359284

CC(C)Cn1c(=O)[nH]c2c(ncn2C)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 7/20 0.39
PDE1B Q01064 7/20 0.39
PDE1C Q14123 7/20 0.39
PDE2A O00408 5/20 0.39
TSHR P16473 3/20 0.39
CFTR P13569 2/20 0.39
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
CYP3A4 P08684 2/20 0.39
PDE5A O76074 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.39
ADORA1 P30542 1/20 0.39
SCN1A P35498 1/20 0.39
PDE6C P51160 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE7A Q13946 1/20 0.39
PDE3A Q14432 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5647 0.77 ADORA2A (0.43) PDE1APDE1BPDE1CPDE2ATSHR
SCHEMBL515776 0.76 ALDH1A1 (0.54) TSHRCYP3A4MAPK1ADORA1ADORA2A
SCHEMBL9031171 0.74 PDE4A (0.35) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL169145 0.73 KDM4E (0.41) PDE1APDE1BPDE1CPDE2ATSHR
SCHEMBL27620150 0.73 CYP3A4 (0.40) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL9885811 0.73 KDM4E (0.48) PDE1APDE1BPDE1CPDE2ATSHR
SCHEMBL18991108 0.71 HSP90B1 (0.46) CYP3A4CYP1A2MAPK1LMNAMAPT
SCHEMBL2462137 0.71 PDE4A (0.69) PDE1APDE1BPDE1CPDE4APDE4B
SCHEMBL13111707 0.69 PDE1A (0.49) PDE1APDE1BPDE1CPDE2ATSHR
SCHEMBL16359618 0.68 ADORA2A (0.45) PDE4APDE4BPDE4CPDE4DCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999026657-A1 INHIBITORS OF NITRIC OXIDE SYNTHASE MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 1999-06-03 WO disclosed