SCHEMBL8364923

SCHEMBL8364923

O=C1CCC(CCO)(c2ccc(F)c(F)c2)CN1Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.54
TACR2 P21452 2/20 0.49
TACR3 P29371 2/20 0.49
CCR5 P51681 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8485199 0.85 TACR1 (0.44) TACR1TACR2TACR3
SCHEMBL8366723 0.83 TACR1 (0.49) TACR1TACR2TACR3
SCHEMBL8203185 0.80 TACR1 (0.68) TACR1TACR2TACR3CCR5
SCHEMBL4630131 0.77 HSD11B1 (0.36) TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8366693 0.77 TACR1 (0.59) TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8364665 0.76 TACR1 (0.56) TACR1TACR2TACR3CCR5
SCHEMBL8483549 0.75 TACR1 (0.56) TACR1TACR2TACR3
SCHEMBL8347511 0.74 KDM4E (0.45) TACR1TACR2TACR3CCR5
SCHEMBL7956540 0.74 CCR5 (0.58) TACR1TACR2TACR3CCR5
SCHEMBL8991919 0.74 TACR1 (0.42) TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965580-A TREATMENT OF SUBSTANCE P- AND NEUROKININ-DEPENDENT DISORDERS SANOFI (FR) 1999-10-12 US disclosed