SCHEMBL8366248

SCHEMBL8366248

CC1(C)CCC(C)(C)c2cc(C3CC3C=O)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 14/20 0.47
RARB P10826 13/20 0.47
RARG P13631 13/20 0.47
RARA P10276 7/20 0.41
CYP26A1 O43174 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
GMNN O75496 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
NFKB1 P19838 1/20 0.39
CYP2C19 P33261 1/20 0.39
THPO P40225 1/20 0.39
MTOR P42345 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8364733 1.00 RXRA (0.47) RXRARARBRARGRARACYP26A1
SCHEMBL7878388 0.80 RXRA (0.48) RXRARARBRARGRARACYP26A1
SCHEMBL18573596 0.78 RXRA (0.43) RXRARARBRARGRARACYP26A1
SCHEMBL6758724 0.77 RARB (0.43) RXRARARBRARGRARA
SCHEMBL727074 0.76 RXRA (0.78) RXRARARBRARGRARARXRB
SCHEMBL8364736 0.76 RXRA (0.78) RXRARARBRARGRARARXRB
SCHEMBL4895819 0.76 RXRA (0.78) RXRARARBRARGRARARXRB
SCHEMBL8366242 0.76 RXRA (0.78) RXRARARBRARGRARARXRB
SCHEMBL15886820 0.76 RXRA (0.78) RXRARARBRARGRARARXRB
SCHEMBL727073 0.76 RXRA (0.78) RXRARARBRARGRARARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775103-B1 RETINOIC ACID X-RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 1999-06-09 EP disclosed
US-5801253-A Retinoic acid X-receptor ligands HOFFMANN-LA ROCHE INC. (US) 1998-09-01 US disclosed
WO-1996039374-A1 2,4-PENTADIENOIC ACID DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-12-12 WO disclosed