SCHEMBL8369705

SCHEMBL8369705

O=CNc1nc(Br)c2[nH]cnc2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 2/20 0.37
DPP4 P27487 1/20 0.37
ALDH1A1 P00352 1/20 0.36
PNP P00491 1/20 0.36
GDA Q9Y2T3 2/20 0.35
PDPK1 O15530 1/20 0.35
PRKACA P17612 2/20 0.35
XDH P47989 1/20 0.34
CDK2 P24941 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CHEK1 O14757 1/20 0.34
AURKA O14965 1/20 0.34
CHEK2 O96017 1/20 0.34
ABL1 P00519 1/20 0.34
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
CDK1 P06493 1/20 0.34
LYN P07948 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28141583 0.82 XDH (0.41) NEK2DPP4ALDH1A1XDHCDK2
SCHEMBL6551675 0.81 DPP4 (0.56) NEK2DPP4ALDH1A1PNPGDA
SCHEMBL28387743 0.81 PDPK1 (0.54) NEK2DPP4ALDH1A1PNPGDA
SCHEMBL8369704 0.75 MEN1 (0.32)
Acetic Acid SCHEMBL7594624 0.74 DPP4 (0.48) NEK2DPP4GDAXDHCDK2
SCHEMBL533603 0.71 PDPK1 (0.44) DPP4ALDH1A1PNPGDAPDPK1
SCHEMBL27337868 0.70 CDK2 (0.54) NEK2ALDH1A1CDK2HSD17B10CDK1
SCHEMBL355362 0.68 PDPK1 (0.66) DPP4GDAPDPK1PRKACACDK2
SCHEMBL1901598 0.68 GDA (0.60) PNPGDAXDHPOLA1
Lithium SCHEMBL30870625 0.67 GDA (0.58) PNPGDAXDHPOLA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543095-B1 Method for producing 2-amino-6-halogenopurine and synthesis of an intermediate therefore SUMIKA FINE CHEMICALS CO LTD (JP) 1999-01-20 EP disclosed
US-5440037-A Method for production of 2-amino-6-halogenopurine derivatives SUMIKA FINE CHEMICALS CO., LTD. (JP) 1995-08-08 US disclosed
US-5391733-A Synthesis intermediates for 2-amino-6-halogenopurines SUMIKA FINE CHEMICALS CO., LTD. (JP) 1995-02-21 US disclosed
US-5389637-A 2-formylamino-6-halogenopurine SUMIKA FINE CHEMICALS CO., LTD. (JP) 1995-02-14 US disclosed
EP-0543095-A2 Method for producing 2-amino-6-halogenopurine and synthesis intermediate therefor SUMIKA FINE CHEMICALS Co., Ltd. (JP) 1993-05-26 EP disclosed