SCHEMBL837009

SCHEMBL837009

O=C(Cl)C(Cl)c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALPG P10696 1/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
HTT P42858 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3070290 0.82 HDAC3 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1511329 0.80 HDAC3 (0.44) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1395758 0.80 HDAC3 (0.44) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL11336506 0.79 BRD4 (0.47) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL5684986 0.79 HDAC3 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL11753976 0.78 CES2 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1398583 0.78 HDAC3 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL27845968 0.77 HDAC3 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8657004 0.77 SMN1; SMN2 (0.42) CES2CES1ALDH1A1LMNASMN1; SMN2
SCHEMBL9558442 0.77 CES2 (0.45) HDAC4HDAC7HDAC5CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041316-A TAM family kinase/and CSF1R kinase inhibitor and application thereof 南京药捷安康生物科技有限公司 2019-07-23 CN disclosed
CN-109575018-A A kind of anti-infective compounds 韩国巴斯德研究所 2019-04-05 CN disclosed
CN-106103439-B 2,7- diaza spiro [3.5] nonane compound 瑞敏德股份有限公司 2019-03-08 CN disclosed
CN-109414421-A The inhibitor and its application method of indole amine 2,3-dioxygenase 百时美施贵宝公司 2019-03-01 CN disclosed
CN-108440370-A Inhibitors of viral replication 鲁汶天主教大学 2018-08-24 CN disclosed
CN-104024223-B Inhibitors of viral replication 鲁汶天主教大学 2018-07-24 CN disclosed
CN-108191746-A A kind of novel hydroxyl pyridine compounds and preparation method and application 暨南大学 2018-06-22 CN disclosed
CN-107820492-A Pyridin-3-yl acetic acid derivatives as inhibitors of HIV replication VIIV保健英国第五有限公司 2018-03-20 CN disclosed
CN-103980219-B A kind of novel bacterial quorum sensing regulator and medical application thereof 中国人民解放军军事医学科学院毒物药物研究所 2016-12-28 CN disclosed
CN-106103439-A 2,7 diaza spiros [3.5] nonane compound 瑞敏德股份有限公司 2016-11-09 CN disclosed
CN-101128199-A Monocyclic heterocycles as kinase inhibitors BRISTOL MYERS SQUIBB CO (US) 2008-02-20 CN disclosed
CN-101005843-A Pyrrolotriazine kinase inhibitors BRISTOL MYERS SQUIBB CO (US) 2007-07-25 CN disclosed
CN-1993130-A Processes and intermediates useful for preparing fused heterocyclic kinase inhibitors BRISTOL MYERS SQUIBB CO (US) 2007-07-04 CN disclosed
WO-2007017261-A1 XANTHINE DERIVATIVES AS SELECTIVE HM74A AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed
WO-2007017262-A1 XANTHINE DERIVATIVES AS SELECTIVE HM74A AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed
CN-1671386-A Substituted anilinic piperidines as MCH selective antagonists LUNDBECK & CO AS H (DK) 2005-09-21 CN disclosed
CN-1668300-A Spirocyclic piperidines as MCH1 antagonists and uses thereof LUNDBECK & CO AS H (DK) 2005-09-14 CN disclosed
CN-1642600-A 1,2-dihydropyrazol-3-ones which controls inflammatory cytokines PROCTER & GAMBLE (US) 2005-07-20 CN disclosed
US-5032588-A Non-steroidal antiinflammatory ABBOTT LABORATORIES (US) 1991-07-16 US disclosed
WO-1991008744-A1 THIAZOLE LIPOXYGENASE-INHIBITING COMPOUNDS DERIVED FROM NON-STEROIDAL ANTIINFLAMMATORY CARBOXYLIC ACIDS ABBOTT LABORATORIES (US) 1991-06-27 WO disclosed