SCHEMBL9558442

SCHEMBL9558442

O=C(Cl)C(Cl)c1cc(F)cc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.45
CES1 P23141 4/20 0.45
MDM2 Q00987 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35
HDAC4 P56524 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HCAR1 Q9BXC0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10441312 0.82 CES2 (0.45) CES2CES1MDM2CA12CA1
SCHEMBL5504134 0.80 CES2 (0.44) CES2CES1MDM2CA12CA1
SCHEMBL7287698 0.80 CES2 (0.44) CES2CES1MDM2CA12CA1
SCHEMBL9670798 0.79 HDAC4 (0.51) CES2CES1HDAC4HDAC7HDAC5
SCHEMBL837009 0.77 HDAC3 (0.45) CES2CES1CA1HDAC4HDAC7
SCHEMBL8820615 0.74 TPMT (0.41) HCAR1
SCHEMBL28175905 0.73 TPMT (0.39) HCAR1
SCHEMBL1398788 0.72 CES2 (0.38) CES2CES1MDM2HDAC4HDAC7
SCHEMBL28550048 0.71 APP (0.41) CES2CES1MDM2SLC6A3
SCHEMBL28274632 0.70 CES2 (0.46) CES2CES1MDM2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101951912-A Treatment of post-traumatic stress disorder SYNOSIA THERAPEUTICS 2011-01-19 CN disclosed
CN-101198333-A Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER PHARMACEUTICALS CORP (US) 2008-06-11 CN disclosed
CN-1022913-C Herbicidal compositions containing new pyrrolidine derivative and its preparing method MITSUI TOATSU CHEMICALS (JP) 1993-12-01 CN disclosed
EP-0387869-B1 4-ETHYL-3-(SUBSTITUTED PHENYL)-1-(3-TRIFLUOROMETHYL-PHENYL)-2-PYRROLIDINONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USE THEREOF, HERBICIDAL COMPOSITIONS CONTAINING THEM MITSUI TOATSU CHEMICALS, Inc. (JP) 1993-07-21 EP disclosed
US-5131947-A 4-ETHYL-3-(SUBSTITUTED PHENYL)-1-(3-TRIFLUOROMETHYLPHENYL)-2-PYRROLIDINONE DERIVATIVES, HERBICIDAL COMPOSITIONS CONTAINING THEM AND USE THEREOF MITSUI TOATSU CHEMICALS INCORPORATED (JP) 1992-07-21 US disclosed
CN-1045581-A 4-ethyl-3-(substituted-phenyl)-1-(3-trifluoromethyl)-2-Pyrrolidone derivative, its preparation method contains the herbicidal composition of this derivative as activeconstituents MITSUI TOATSU CHEMICALS (JP) 1990-09-26 CN disclosed
EP-0387869-A2 4-Ethyl-3-(substituted phenyl)-1-(3-trifluoromethyl-phenyl)-2-pyrrolidinone derivatives, processes for the preparation and use thereof, herbicidal compositions containing them MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-09-19 EP disclosed