SCHEMBL8370748

SCHEMBL8370748

Nc1cccc(CNc2nccc3ccccc23)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.52
RPS6KB1 P23443 1/20 0.52
ELANE P08246 1/20 0.49
EGFR P00533 2/20 0.48
KLKB1 P03952 1/20 0.47
KLK1 P06870 1/20 0.47
IGF1R P08069 1/20 0.46
APP P05067 7/20 0.45
GRM4 Q14833 1/20 0.45
ROCK1 Q13464 2/20 0.43
F12 P00748 1/20 0.42
PLAU P00749 1/20 0.42
NCF1 P14598 1/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
BACE1 P56817 1/20 0.42
WNT3A P56704 1/20 0.42
UTS2R Q9UKP6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31098952 0.84 EGFR (0.57) EGFRAPPGRM4WNT3AUTS2R
SCHEMBL6477749 0.84 EGFR (0.57) EGFRAPPGRM4WNT3AUTS2R
Methane SCHEMBL9378754 0.82 EGFR (0.55) EGFRAPPGRM4WNT3AUTS2R
SCHEMBL10055014 0.82 WNT3A (0.54) EGFRAPPGRM4WNT3AUTS2R
SCHEMBL27990386 0.78 EGFR (0.71) AURKARPS6KB1ELANEEGFRAPP
SCHEMBL9927462 0.77 CYP1A2 (0.56) EGFR
SCHEMBL7127641 0.77 AHR (0.58) EGFRF12PLAUNCF1NOS3
SCHEMBL10055013 0.75 WNT3A (0.48) EGFRGRM4WNT3AUTS2R
SCHEMBL7122983 0.73 AURKA (0.43) AURKARPS6KB1GRM4
SCHEMBL509566 0.72 EGFR (0.64) AURKARPS6KB1EGFRIGF1RAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11130750-A None JP disclosed
JP-H11130750-A NOVEL DERIVATIVE FUJISAWA PHARMACEUT CO LTD 1999-05-18 JP disclosed