Methane

Methane

SCHEMBL9378754

C.c1ccc(CNc2nccc3ccccc23)cc1

nearest known ligand 0.66

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.55
GALR3 O60755 2/20 0.55
NR2F2 P24468 2/20 0.55
RAB9A P51151 1/20 0.55
UTS2R Q9UKP6 1/20 0.55
LMNA P02545 2/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
RAD52 P43351 2/20 0.53
KMT2A Q03164 5/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
PKM P14618 1/20 0.51
UBE2N P61088 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
RCE1 Q9Y256 1/20 0.51
PDE5A O76074 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6477749 0.98 EGFR (0.57) EGFRGALR3NR2F2RAB9AUTS2R
SCHEMBL31098952 0.98 EGFR (0.57) EGFRGALR3NR2F2RAB9AUTS2R
SCHEMBL10055014 0.93 WNT3A (0.54) EGFRGALR3NR2F2RAB9AUTS2R
SCHEMBL10055013 0.86 WNT3A (0.48) EGFRGALR3NR2F2RAB9AUTS2R
SCHEMBL9927462 0.84 CYP1A2 (0.56) EGFRRAB9ALMNATSHRMAPK1
SCHEMBL509566 0.82 EGFR (0.64) EGFRNR2F2MAPK1KMT2AKDM4E
SCHEMBL8370748 0.82 AURKA (0.52) EGFRUTS2RAPPGRM4WNT3A
SCHEMBL9374978 0.82 RAB9A (0.59) EGFRRAB9AUTS2RLMNAMAPK1
SCHEMBL29647714 0.82 HDAC6 (0.62)
SCHEMBL19631286 0.82 HDAC6 (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0393926-B1 1-Aminoisoquinoline derivatives SMITHKLINE BEECHAM INTERCREDIT (NL) 1994-09-21 EP disclosed
US-5200417-A Administering to inhibait gastric acid secretion in mammals SMITHKLINE BEECHAM INTERCREDIT B.V. (GB) 1993-04-06 US disclosed
EP-0393926-A1 1-Aminoisoquinoline derivatives SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1990-10-24 EP disclosed