SCHEMBL8370834

SCHEMBL8370834

CC(=O)N(c1ccc(C#N)cc1)c1c(NC(C)C)c(=O)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.52
PLK4 O00444 1/20 0.52
DAPK3 O43293 1/20 0.52
ROCK2 O75116 1/20 0.52
CHEK2 O96017 1/20 0.52
PIM1 P11309 1/20 0.52
FLT4 P35916 1/20 0.52
KDR P35968 1/20 0.52
GSK3A P49840 1/20 0.52
GSK3B P49841 1/20 0.52
RPS6KA3 P51812 1/20 0.52
PRKX P51817 1/20 0.52
PLK1 P53350 1/20 0.52
CSNK1G2 P78368 1/20 0.52
PRKCZ Q05513 1/20 0.52
ROCK1 Q13464 1/20 0.52
PRKG1 Q13976 1/20 0.52
CDC42BPA Q5VT25 1/20 0.52
AURKB Q96GD4 1/20 0.52
PLK3 Q9H4B4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8369527 0.90 CDC7 (0.53) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8369802 0.88 CDC7 (0.48) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8369762 0.88 PLK1 (0.69) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8369755 0.88 PLK1 (0.69) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8870428 0.86 ROCK1 (0.49) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8870420 0.86 ROCK1 (0.49) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8369736 0.85 DAPK3 (0.44) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8369737 0.85 DAPK3 (0.44) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8369858 0.78 MGLL (0.43) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8371877 0.77 PLK1 (0.56) CDC7PLK4DAPK3ROCK2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0796243-B1 DIAMINOCYCLOBUTENE-3,4-DIONES AMERICAN HOME PROD (US) 1999-01-27 EP claimed
EP-0796243-A1 DIAMINOCYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1997-09-24 EP claimed
WO-1996015103-A1 DIAMINOCYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1996-05-23 WO claimed
US-5464867-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-07 US claimed
EP-0796243-B1 DIAMINOCYCLOBUTENE-3,4-DIONES AMERICAN HOME PROD (US) 1999-01-27 EP disclosed
US-5536741-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-16 US disclosed
US-5536731-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-16 US disclosed
US-5530025-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-06-25 US disclosed