SCHEMBL8374471

SCHEMBL8374471

O=S(=O)(Nc1c(F)cccc1F)c1nc2sccn2n1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.36
MAPT P10636 3/20 0.36
TP53 P04637 2/20 0.36
MAPK1 P28482 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
ALOX15 P16050 1/20 0.36
GAA P10253 2/20 0.35
SMN1; SMN2 Q16637 4/20 0.34
PKM P14618 2/20 0.34
HPGD P15428 1/20 0.34
USP2 O75604 2/20 0.34
ALDH1A1 P00352 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10561074 0.81 SMN1; SMN2 (0.43) MAPTTP53KMT2AGAASMN1; SMN2
SCHEMBL7851317 0.76 JAK2 (0.38) MAPK1KMT2APOLBGAASMN1; SMN2
Flumetsulam SCHEMBL54906 0.74 TSHR (0.40) MAPK1KMT2AGAASMN1; SMN2USP2
SCHEMBL10660778 0.74 HPGD (0.40) LMNASMN1; SMN2HPGDALDH1A1
SCHEMBL7851017 0.73 ACLY (0.37)
Flumetsulam SCHEMBL20723449 0.73 TSHR (0.39) MAPK1KMT2AGAASMN1; SMN2USP2
Flumetsulam SCHEMBL20723426 0.73 TSHR (0.39) MAPK1KMT2AGAASMN1; SMN2USP2
SCHEMBL9375954 0.72 GAA (0.33) MAPK1KMT2AGAASMN1; SMN2USP2
SCHEMBL7851696 0.72 GAA (0.45) MAPTMAPK1KMT2APOLBGAA
SCHEMBL27747678 0.72 KMT2A (0.40) MAPK1KMT2AMEN1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5484760-A AMIDES MONSANTO COMPANY (US) 1996-01-16 US claimed
EP-0565593-A1 REDUCING PESTICIDAL INTERACTIONS IN CROPS MONSANTO COMPANY (US) 1993-10-20 EP claimed
EP-0562015-A1 SAFENED HERBICIDAL SULFONAMIDE COMPOSITIONS MONSANTO COMPANY (US) 1993-09-29 EP claimed
WO-1992011761-A1 REDUCING PESTICIDAL INTERACTIONS IN CROPS MONSANTO COMPANY (US) 1992-07-23 WO claimed
WO-1992010098-A1 SAFENED HERBICIDAL SULFONAMIDE COMPOSITIONS MONSANTO COMPANY (US) 1992-06-25 WO claimed
US-4795483-A THIAZOLO-TRIAZOLE SULFONAMIDES SCHERING AGROCHEMICALS (GB) 1989-01-03 US claimed
EP-0244098-A2 Thiazolotriazole herbicides SCHERING AGROCHEMICALS LIMITED (GB) 1987-11-04 EP claimed
EP-0565593-B1 REDUCING PESTICIDAL INTERACTIONS IN CROPS MONSANTO CO (US) 1999-03-03 EP disclosed
US-5484760-A AMIDES MONSANTO COMPANY (US) 1996-01-16 US disclosed
EP-0565593-A1 REDUCING PESTICIDAL INTERACTIONS IN CROPS MONSANTO COMPANY (US) 1993-10-20 EP disclosed
EP-0562015-A1 SAFENED HERBICIDAL SULFONAMIDE COMPOSITIONS MONSANTO COMPANY (US) 1993-09-29 EP disclosed
WO-1992011761-A1 REDUCING PESTICIDAL INTERACTIONS IN CROPS MONSANTO COMPANY (US) 1992-07-23 WO disclosed
WO-1992010098-A1 SAFENED HERBICIDAL SULFONAMIDE COMPOSITIONS MONSANTO COMPANY (US) 1992-06-25 WO disclosed
US-4795483-A THIAZOLO-TRIAZOLE SULFONAMIDES SCHERING AGROCHEMICALS (GB) 1989-01-03 US disclosed
EP-0244098-A2 Thiazolotriazole herbicides SCHERING AGROCHEMICALS LIMITED (GB) 1987-11-04 EP disclosed