SCHEMBL8375768

SCHEMBL8375768

OCCC(Cl)(Cl)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
CYP1A2 P05177 2/20 0.43
TDP1 Q9NUW8 1/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2C9 P11712 1/20 0.37
KIF11 P52732 5/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KCNN4 O15554 1/20 0.35
HIF1A Q16665 1/20 0.34
RECQL P46063 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8376477 0.86 TSHR (0.42) TSHRCYP1A2TDP1CYP2C19CYP2C9
SCHEMBL8379857 0.81 TSHR (0.46) TSHRCYP1A2CYP2C19CYP2C9KIF11
SCHEMBL7409166 0.80 TSHR (0.50) TSHRCYP1A2TDP1CYP2C19CYP2C9
SCHEMBL28790232 0.79 TSHR (0.44) TSHRCYP1A2TDP1CYP2C19CYP2C9
SCHEMBL11814132 0.78 TSHR (0.48) TSHRCYP1A2CYP2C19CYP2C9KIF11
SCHEMBL2102354 0.78 TSHR (0.48) TSHRCYP1A2CYP2C19CYP2C9KIF11
SCHEMBL9618238 0.76 KIF11 (0.50) TSHRCYP1A2CYP2C19CYP2C9KIF11
SCHEMBL6680627 0.76 TSHR (0.46) TSHRCYP1A2CYP2C19CYP2C9KIF11
SCHEMBL27491062 0.76 TSHR (0.46) TSHRCYP1A2TDP1CYP2C19CYP2C9
SCHEMBL8166179 0.76 CYP1A2 (0.48) TSHRCYP1A2CYP2C19KIF11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108379686-B Non-packaging syringe assembly with sterilizable fluid path 贝克顿·迪金森公司 2020-10-16 CN disclosed
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed