SCHEMBL8375787

SCHEMBL8375787

NC(O)(CCc1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KIF11 P52732 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
CYP2A6 P11509 1/20 0.43
HTR2A P28223 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
GRM2 Q14416 1/20 0.42
GRM3 Q14832 1/20 0.42
CES1 P23141 1/20 0.42
KCNN4 O15554 1/20 0.41
MAOA P21397 3/20 0.40
CHRM3 P20309 2/20 0.40
MAOB P27338 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28681602 0.80 SMN1; SMN2 (0.48) CYP1A2CYP2C9CYP2C19SMN1; SMN2CYP2A6
SCHEMBL27491063 0.79 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19KIF11TDP1
Hydrochloric Acid SCHEMBL8670716 0.78 MAOB (0.46) CYP1A2CYP2C9CYP2C19SMN1; SMN2CYP2A6
SCHEMBL4779153 0.78 CYP2C9 (0.50) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2
SCHEMBL2067595 0.78 CYP1A2 (0.61) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2
SCHEMBL11264802 0.78 SMN1; SMN2 (0.46) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2
SCHEMBL28065368 0.78 SMN1; SMN2 (0.52) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2
SCHEMBL2067126 0.78 CYP1A2 (0.61) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2
SCHEMBL4750696 0.78 KCNN4 (0.44) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2
SCHEMBL82460 0.78 CYP1A2 (0.61) CYP1A2CYP2C9CYP2C19KIF11SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104016877-A Acetylaniline compounds and application thereof in preparation of mirabegron NANJING HAIRONG PHARMACEUTICAL TECHNOLOGY CO LTD 2014-09-03 CN disclosed
US-5919990-A Reclamation of bisphenol tars as feedstock in the synthesis of aminophenylhydroxphenylalkanes GENERAL ELECTRIC COMPANY (US) 1999-07-06 US disclosed
EP-0837051-A2 Synthesis of aminophenylhydroxyphenylalkanes form bisphenol tars GENERAL ELECTRIC COMPANY (US) 1998-04-22 EP disclosed
EP-0052963-B1 SECONDARY AMINES BEECHAM GROUP PLC (GB) 1985-02-20 EP disclosed