SCHEMBL8375794

SCHEMBL8375794

[CH2]CC(OCCCCCC)c1cccc2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.43
CNR1 P21554 2/20 0.42
CNR2 P34972 2/20 0.42
CYP2C9 P11712 2/20 0.40
HTR1B P28222 4/20 0.39
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR1D P28221 2/20 0.37
PLA2G2D Q9UNK4 1/20 0.37
FAAH O00519 1/20 0.37
MGLL Q99685 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16058112 0.82 CNR1 (0.44) AOC3CNR1CNR2CYP2C9HTR1B
SCHEMBL25329203 0.81 CASP1 (0.36) KDM4EKMT2AALDH1A1
SCHEMBL7931404 0.80 KDM4E (0.44) AOC3CNR1CNR2CYP2C9HTR1B
SCHEMBL6756012 0.77 NPC1 (0.43) ALDH1A1
SCHEMBL8375755 0.77 AOC3 (0.62) AOC3CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL8377421 0.77 KDM4E (0.42) CNR1CNR2CYP2C9KDM4EKMT2A
SCHEMBL28188122 0.77 KDM4E (0.42) CNR1CNR2CYP2C9KDM4EKMT2A
SCHEMBL28188781 0.77 KDM4E (0.42) CNR1CNR2CYP2C9KDM4EKMT2A
SCHEMBL28188830 0.77 KDM4E (0.42) CNR1CNR2CYP2C9KDM4EKMT2A
SCHEMBL28188829 0.77 KDM4E (0.42) CNR1CNR2CYP2C9KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
CN-1216986-A Isoxazole derivatives SANKYO CO (JP) 1999-05-19 CN disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed