SCHEMBL8375805

SCHEMBL8375805

OC(CF)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.58
KDM4E B2RXH2 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
AOC3 Q16853 5/20 0.52
RIPK1 Q13546 1/20 0.48
BCAT2 O15382 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TSHR P16473 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25202788 1.00 LMNA (0.58) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL23363771 1.00 LMNA (0.58) LMNAKDM4EL3MBTL1AOC3RIPK1
Hydrochloric Acid SCHEMBL28216040 0.97 LMNA (0.56) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL28218514 0.81 LMNA (0.50) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL14568664 0.80 RIPK1 (0.55) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL8377394 0.80 RIPK1 (0.55) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL5610567 0.78 RIPK1 (0.53) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL18256215 0.78 RIPK1 (0.53) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL28983014 0.78 LMNA (0.47) LMNAKDM4EL3MBTL1AOC3RIPK1
SCHEMBL3096537 0.78 LMNA (0.64) LMNAKDM4EL3MBTL1AOC3RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103649263-A Direct trifluoromethylation using trifluoromethane UNIV SOUTHERN CALIFORNIA 2014-03-19 CN claimed
US-12545684-B2 CDK2 inhibitors BLUEPRINT MEDICINES CORPORATION (US) 2026-02-10 US disclosed
US-20240383902-A1 CDK2 INHIBITORS BLUEPRINT MEDICINES CORPORATION 2024-11-21 US disclosed
US-11999717-B2 Triazole carbamate pyridyl sulfonamides as LPA receptor antagonists and uses thereof GILEAD SCIENCES, INC. (US) 2024-06-04 US disclosed
EP-4363423-A1 CDK2 INHIBITORS Blueprint Medicines Corporation (US) 2024-05-08 EP disclosed
US-11970498-B2 CDK2 inhibitors BLUEPRINT MEDICINES CORPORATION (US) 2024-04-30 US disclosed
CN-117897384-A CDK2 inhibitors 缆图药品公司 2024-04-16 CN disclosed
CN-114728168-B Triazole carbamate pyridylsulfonamides as LPA receptor antagonists and their use 吉利德科学公司 2024-04-09 CN disclosed
US-11932648-B2 CDK2 inhibitors BLUEPRINT MEDICINES CORPORATION (US) 2024-03-19 US disclosed
CN-117358275-A Carbon nitride molecular junction catalyst and preparation method and application thereof 深圳大学 2024-01-09 CN disclosed
US-7592486-B2 Anhydrous fluoride salts and reagents and methods for their production BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2009-09-22 US disclosed
CN-101351451-A Polycyclic amino acid derivatives and methods of use thereof LEXICON GENETICS INC (US) 2009-01-21 CN disclosed
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed
EP-0415833-B1 Optically active fluorine-containing alcohol compounds and liquid crystal compounds therefrom SHOWA SHELL SEKIYU (JP) 1996-09-11 EP disclosed
US-5096613-A OPTICALLY ACTIVE FLUORINE-CONTAINING ALCOHOL COMPOUNDS AND LIQUID CRYSTAL COMPOUNDS THEREFROM SHOWA SHELL SEKIYU KABUSHIKI KAISHA (JP) 1992-03-17 US disclosed
EP-0415833-A2 Optically active fluorine-containing alcohol compounds and liquid crystal compounds therefrom Showa Shell Sekiyu Kabushiki Kaisha (JP) 1991-03-06 EP disclosed
US-4861801-A Treatment of depression by using a fluorophenacylamine derivative Lafon, Laboratoire L. (FR) 1989-08-29 US disclosed
US-4835315-A Fluorophenacyl-amine derivatives and application thereof in therapeutics LABORATOIRE L. LAFON (FR) 1989-05-30 US disclosed
EP-0060954-B1 DERIVATIVES OF FLUOROPHENACYL AMINES AND THEIR THERAPEUTIC USE LABORATOIRE L. LAFON Société anonyme dite: (FR) 1984-08-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11932648-B2 CDK2 inhibitors CDK2, CDK20, CDK2AP1 LMNA 2403/4885KDM4E 2160/4885L3MBTL1 2771/4885
US-11999717-B2 Triazole carbamate pyridyl sulfonamides as LPA receptor antagonists and uses thereof LPAR3, LPAR1, LPAR2 LMNA 1879/4885KDM4E 2137/4885L3MBTL1 2693/4885
US-11970498-B2 CDK2 inhibitors CDK2, CDK20, CDK2AP1 LMNA 2403/4885KDM4E 2160/4885L3MBTL1 2771/4885
US-20240383902-A1 CDK2 INHIBITORS CDK2, CDK20, CDK2AP1 LMNA 2403/4885KDM4E 2160/4885L3MBTL1 2771/4885
US-12545684-B2 CDK2 inhibitors CDK2, CDK4, CDK1 LMNA 1435/4885KDM4E 1727/4885L3MBTL1 2557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.