SCHEMBL8375901

SCHEMBL8375901

Cc1ccc(O)c2c3c(n(Cc4ccccc4)c12)CCCC3C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 11/20 0.43
FABP3 P05413 2/20 0.43
PLA2G2A P14555 1/20 0.41
HTR6 P50406 2/20 0.39
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375966 0.89 FABP4 (0.41) FABP4FABP3PLA2G2AHTR6
SCHEMBL8374848 0.89 FABP4 (0.41) FABP4FABP3PLA2G2AHTR6
SCHEMBL6697582 0.87 PLA2G2A (0.44) FABP4FABP3PLA2G2AHTR6
SCHEMBL6129678 0.87 FABP4 (0.43) FABP4FABP3PLA2G2AHTR6
SCHEMBL27844976 0.85 FABP4 (0.39) FABP4FABP3PLA2G2AHTR6
SCHEMBL818322 0.85 PLA2G2A (0.47) PLA2G2A
SCHEMBL29862757 0.85 PLA2G2A (0.47) PLA2G2A
SCHEMBL6129679 0.84 FABP4 (0.38) FABP4FABP3PLA2G2AHTR6
SCHEMBL6691719 0.83 PLA2G2A (0.49) FABP4FABP3PLA2G2AHTR6
SCHEMBL6693186 0.82 PLA2G2A (0.49) PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0952149-A2 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitiors ELI LILLY AND COMPANY (US) 1999-10-27 EP claimed