SCHEMBL8377331

SCHEMBL8377331

CN(C)C(=O)c1cccc2cc3ccccc3cc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
KDM4E B2RXH2 3/20 0.61
GAA P10253 1/20 0.61
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
KEAP1 Q14145 1/20 0.46
POLB P06746 1/20 0.46
GABRA1 P14867 1/20 0.41
GABRB2 P47870 1/20 0.41
PKN1 Q16512 1/20 0.40
PKN2 Q16513 1/20 0.40
HPGD P15428 2/20 0.40
GLA P06280 2/20 0.40
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40
MAPT P10636 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10407111 0.83 NR4A1 (0.59) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL3624238 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EGAAKMT2AKEAP1
SCHEMBL5304396 0.80 KMT2A (0.50) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL7610003 0.79 KDM4E (0.67) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL29875368 0.79 KDM4E (0.67) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL978940 0.79 KDM4E (0.67) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL578683 0.79 KDM4E (0.71) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL29052004 0.78 KDM4E (0.65) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL123193 0.77 ALDH1A1 (0.69) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL29196640 0.77 KDM4E (0.69) ALDH1A1KDM4EGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed